SAQPhysiologyNeurophysiology2002 · Perception and modulation of pain

Question bank · 2002 · Physiology

The same injury does not always hurt the same.
Perception is built in the brain, and adjusted at every synapse on the way.

Show the model answerAttempt it first — that is what makes it stick

How pain is perceived

What earns the marks

TransductionNociceptor free endings; mediators and noxious stimuli open channels; action potentials
TransmissionAδ first pain and C second pain to the dorsal horn
The three neuronesDorsal root ganglion; dorsal horn, crossing to the spinothalamic tract; thalamus to cortex
Two streamsLateral: where and how intense. Medial: how unpleasant
PerceptionA distributed network, the pain matrix, not a single centre; each area's contribution

Read the question: The verb is perceived. An answer that stops at the spinothalamic tract has described transmission. The marks for perception are in what the cortex does with the signal: the sensory and the emotional components, and where each is made.

Pathway

The ascending pathway, in three neurons

Read it from the bottom. The first-order neuron has its cell body in the dorsal root ganglion, outside the cord, and synapses in the dorsal horn. The second-order neuron starts in the dorsal horn, crosses in the cord and ascends on the opposite side. At the brainstem the projection divides: the lateral, neospinothalamic route relays in the ventral posterolateral nucleus (VPL) and reaches the primary somatosensory cortex, which is where and how intense; the medial, paleospinothalamic route passes through the reticular formation and periaqueductal grey to the intralaminar nuclei and on to the cingulate and insula, which is how unpleasant. The third-order neuron runs from thalamus to cortex. From the face the plan is the same, with the first-order cell body in the trigeminal ganglion, the second in the spinal trigeminal nucleus and the third in the ventral posteromedial nucleus.

CortexS1, S2, insula, anterior cingulateThalamusVPL (lateral) and intralaminar (medial)BrainstemReticular formation, periaqueductal greySpinal cordDorsal horn, laminae I, II and VPeripheryFree nerve endings of nociceptorsmidlineDorsal root ganglionfirst-order cell bodyDorsal horncrosses hereReticular formationand PAGVPLIntralaminarS1: locationCingulate, insula: affect123NeospinothalamicPaleospinothalamic
StepWhereWhat happens
TransductionNociceptor: free nerve endings in skin, muscle, joints and visceraNoxious heat, pressure or chemicals, and mediators from injured tissue (K⁺, H⁺, ATP, bradykinin, serotonin), open TRPV1, ASIC and P2X3 channels. The generator potential fires action potentials through voltage-gated Na⁺ channels such as Nav1.8
TransmissionAδ and C fibres; cell body in the dorsal root ganglionAδ, thinly myelinated, 12 to 30 m/s: sharp, localised first pain. C, unmyelinated, 0.5 to 2 m/s: dull, diffuse second pain
First synapseDorsal horn: Aδ to laminae I and V, C to lamina IIGlutamate on AMPA and NMDA receptors, substance P on NK1, onto nociceptive-specific and wide dynamic range neurones. This is the first place the signal is modulated
AscentSecond-order neuroneCrosses in the ventral white commissure within one or two segments and ascends in the contralateral anterolateral quadrant
Lateral streamNeospinothalamic: ventral posterolateral thalamus to primary and secondary somatosensory cortexThe sensory-discriminative component: where the stimulus is, how intense, how long
Medial streamPaleospinothalamic, spinoreticular and spinolimbic: reticular formation, periaqueductal grey, intralaminar thalamus, hypothalamus and amygdalaThe motivational-affective component: unpleasantness, arousal, the autonomic response. Reticular activation also starts descending inhibition

The cortex: a network, not a centre

Functional imaging during acute pain shows a set of areas active together, the pain matrix. Broadly, the somatosensory cortices make the sensory-discriminative component and the limbic and paralimbic areas the affective one.

AreaContribution
Primary somatosensory cortexLocalisation
Secondary somatosensory cortexIntensity, and spatial appreciation
InsulaIntensity, and the pain-related autonomic response
Anterior cingulate cortexResponse selection, attention, affect, appraisal
Prefrontal cortexAffect, emotion, memory, modulation

The two components can be separated. Damage to the prefrontal cortex reduces the ability to judge how severe a pain is, and cingulotomy reduces its emotional component. The anterior cingulate and prefrontal cortex also project back to the periaqueductal grey, which is how perception reaches back down to modulate its own input.

How the perception of pain can be modulated, with examples

What earns the marks

Segmental: the gateAβ input excites an inhibitory interneurone in the substantia gelatinosa. Example: rubbing, TENS
How inhibition worksPresynaptic (less transmitter released) and postsynaptic (hyperpolarisation)
DescendingPAG to rostral ventromedial medulla (serotonin) and locus coeruleus (noradrenaline), to the dorsal horn. Example: PAG stimulation, morphine
Endogenous opioidsEnkephalin, β-endorphin, dynorphin. Example: stress-induced analgesia
Higher centresAttention, expectation, mood. Example: placebo analgesia
Upward modulationPeripheral and central sensitisation. Example: sunburn; wind-up
Drugs at each levelNSAIDs, local anaesthetics, opioids, α2 agonists, ketamine, tricyclics

Read the question: With examples” is half the instruction. Every mechanism named should carry one: rubbing an injury for the gate, stress-induced analgesia for the descending opioid system, placebo for expectation, sunburn for sensitisation.

Read the question: Modulation works in both directions. Hyperalgesia after injury is perception turned up, and the brainstem nuclei that inhibit transmission also contain cells that facilitate it. An answer that treats modulation as analgesia alone is incomplete.

1. At the first synapse: the gate

Circuit

The gate, drawn as a circuit

Solid lines excite (+); dashed lines inhibit (−). Both afferents excite the projection neuron directly. The difference is what each does to the inhibitory interneuron in the substantia gelatinosa: the large Aβ fibre excites it, so touch closes the gate; the small C fibre inhibits it, so a noxious input removes the brake and opens the gate twice over. Descending fibres close it from above, by exciting the interneuron and by inhibiting the projection neuron directly.

PAG, RVM and locus coeruleusDescending+descendingAβ fibrelarge, myelinated, touchC fibresmall, unmyelinated, nociceptive+++SGProjTo the brainspinothalamic tractSG: inhibitory interneuron, substantia gelatinosa (lamina II)Proj: projection neuron

Melzack and Wall (1965) proposed that transmission from the primary afferent to the projection neurone is gated by inhibitory interneurones in the substantia gelatinosa, and that the gate’s position is set by the balance of large- and small-fibre input.

InputEffect on the inhibitory interneuroneGateExample
Aβ: touch, pressure, vibrationExcites itClosesRubbing a bumped elbow; transcutaneous electrical nerve stimulation; spinal cord stimulation
Aδ and C: nociceptiveInhibits itOpensThe noxious input itself
Descending fibresExcite it, and inhibit the projection neurone directlyClosesThe route by which descending control, below, acts on the gate

Two places to inhibit the same synapse

An inhibitory transmitter is released in the dorsal horn: opioid peptides, GABA or glycine from interneurones, or noradrenaline and serotonin from descending fibres.
Presynaptic
On the nociceptor's central terminal. Opioid and GABA-B receptors reduce Ca²⁺ entry, so less glutamate and substance P are released.
Postsynaptic
On the projection neurone. Opioids open K⁺ channels and GABA-A receptors open Cl⁻ channels: the cell hyperpolarises.
The same afferent input produces less transmission, so less reaches the cortex to be perceived.
About 75% of dorsal horn opioid receptors are presynaptic.

2. From the brainstem: descending control

The descending pathway, from higher centres to the dorsal horn

Higher centres
Anterior cingulate and prefrontal cortex, hypothalamus and amygdala project to the midbrain; ascending nociceptive fibres send collaterals there too.
Periaqueductal grey
Opioids inhibit its tonically active GABAergic neurones, releasing its output from inhibition.

Brainstem relays

Rostral ventromedial medulla
Including the nucleus raphe magnus. Serotonergic.
Locus coeruleus
Noradrenergic, acting through spinal α2 adrenoceptors.
Dorsal horn
Axons descend in the dorsolateral funiculus to laminae I and II.
Less transmission: presynaptic inhibition, excitation of enkephalin interneurones, and direct postsynaptic inhibition.
  • Example: electrical stimulation of the periaqueductal grey produces profound analgesia, and naloxone reverses it, so endogenous opioids are part of the circuit.
  • Two directions: in the rostral ventromedial medulla, off cells inhibit dorsal horn transmission and on cells facilitate it. Descending control can turn perception up as well as down.

3. The endogenous opioids

PeptideEndogenous agonist at
Enkephalinsδ
β-endorphinµ
Dynorphinsκ

All act through Gi/Go-coupled receptors: adenylyl cyclase is inhibited, voltage-gated Ca²⁺ channels close, and inwardly rectifying K⁺ channels open. The effect is the same cell-level inhibition wherever the receptor is, in the periaqueductal grey, the dorsal horn, or on peripheral terminals in inflamed tissue.

4. From higher centres: stress, attention and expectation

InfluenceExampleMechanism
StressSoldiers wounded in battle often feel little pain until the fighting is overStress-induced analgesia. β-endorphin shares its precursor with ACTH; mice unable to make β-endorphin lose naloxone-reversible stress-induced analgesia
ExpectationPlacebo analgesiaActs on the same brain regions as an opioid, presumably by releasing endogenous opioids
Attention, anxiety, moodThe same injury hurts differently in different people and circumstancesCortical and limbic projections to the periaqueductal grey set the descending system

5. Turning perception up: sensitisation

LevelExampleMechanism
PeripheralSunburnt skin is more sensitive to pain than normal skin: primary hyperalgesiaMediators such as prostaglandins and bradykinin lower the nociceptor's threshold; silent nociceptors are recruited
CentralTenderness in uninjured skin around a wound: secondary hyperalgesia and allodyniaRepeated C-fibre input removes the Mg²⁺ block of the NMDA receptor: wind-up, lower threshold and larger receptive fields in the dorsal horn
Descending facilitationOn cells of the rostral ventromedial medullaFiring just before a withdrawal response, they facilitate dorsal horn transmission

6. Drugs and techniques, each acting at a named step

Step modulatedExample
Peripheral sensitisation by prostaglandinsNSAIDs
Transduction and conduction through Na⁺ channelsLocal anaesthetics
Presynaptic and postsynaptic inhibition in the dorsal horn; the periaqueductal greyOpioids
Spinal α2 adrenoceptors, the target of descending noradrenalineClonidine, dexmedetomidine
The NMDA receptor behind wind-upKetamine
Descending serotonin and noradrenalineTricyclic antidepressants such as amitriptyline
Large-fibre input at the gateTranscutaneous electrical nerve stimulation
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