SAQPharmacologyInhalational agentsMAC, Meyer-Overton and speed of onset

Question bank · Pharmacology

Potency is a partial pressure in the alveolus.
Speed of onset is how quickly the alveolus gets there.

Show the model answerAttempt it first — that is what makes it stick
a

3 marks

MAC, its variants, and the Meyer-Overton hypothesis

Three things in one part: a definition with its conditions, the variants with the end point each one prevents, and the correlation that links MAC to lipid solubility.

What earns the marks3 marks

The definitionAlveolar concentration, steady state, 1 atmosphere, standard surgical stimulus, movement, 50% of subjects
What it measuresPotency: the ED50, and really a partial pressure
The variantsMAC-awake, MAC-BAR, MAC for intubation, MAC95, each with its end point
Meyer-OvertonPotency rises with lipid solubility: MAC × oil:gas coefficient is roughly constant
Its limitsA correlation, not the mechanism

Read the question: “Its variant” asks for the variants by name and by end point. MAC-awake and MAC-BAR written as bare labels say nothing about what each one prevents, which is the only thing that distinguishes them.

  • Steady state matters because only then does the alveolar partial pressure equal the partial pressure in the central nervous system.
  • The immobility it measures is mediated mainly in the spinal cord: decerebration does not change it.
  • MAC varies only 10 to 15% between individuals, and MAC values of different inhaled agents are additive: 0.5 MAC of nitrous oxide with 0.5 MAC of isoflurane behaves as 1 MAC.

The variants

VariantEnd point prevented in 50%Relation to MAC
MAC-awakePerceptive awareness: consciousnessAbout 0.34 × MAC for the potent volatile agents; about 0.7 × MAC for nitrous oxide
MAC-BARThe sympathetic response to incision: a rise in heart rate or mean arterial pressure of more than 15%Reduced by opioids, with a ceiling
MAC for tracheal intubationMovement in response to tracheal intubationThe highest of the stimulus-specific values: intubation is a stronger stimulus than incision
MAC95Movement at incision in 95% of subjectsAbout 1.3 × MAC, because the dose-response curve is steep

MAC-awake lying well below MAC is what makes an ED50 usable at all: a surgeon may tolerate movement in half of patients, but awareness in half would not be acceptable. Some texts give MAC-awake as about half of MAC; the point that carries the mark is that it is a fraction of MAC, and a larger fraction for nitrous oxide.

The relationship with the Meyer-Overton hypothesis

Meyer and Overton observed, independently, that the potency of an anaesthetic rises with its lipid solubility, measured as the oil:gas partition coefficient. Because potency is the reciprocal of MAC, a plot of log MAC against log oil:gas coefficient is a straight line with a negative slope, and the product of the two is roughly constant.

AgentOil:gas coefficientMAC (%)MAC × oil:gas
Halothane2240.75168
Enflurane981.63160
Isoflurane981.17115
Sevoflurane551.899
Desflurane18.76.6123
Nitrous oxide1.4104146

Across a 160-fold range of oil:gas coefficients, the product stays between 99 and 168. One standard text uses 150 as the average, so an estimated MAC is 150 divided by the oil:gas coefficient. The correlation is a line of best fit, not an identity: enflurane and isoflurane share an oil:gas coefficient of 98 and have different MACs.

b

3 marks

Factors affecting MAC

Organise by direction: what raises MAC, what lowers it, and what leaves it unchanged. A list without a direction beside each factor has outlined nothing.

What earns the marks3 marks

Direction for every factorIncrease, decrease, or no change
PhysiologicalAge, temperature, pregnancy
PharmacologicalDrugs that raise or lower central catecholamines; opioids, sedatives, α2 agonists, alcohol, other anaesthetics
PathologicalSodium, severe hypoxaemia and hypotension
No changeSex, duration, PaCO2 across a wide range, potassium

Read the question: The stem is about a 50-year-old. Age is the factor that applies to this patient, and saying so is the difference between an outline and a list copied from a table.

Increase MACDecrease MAC
AgeInfancyIncreasing age, about 6% per decade; the neonatal period
TemperatureHyperthermiaHypothermia
PregnancyPregnancy, by nearly 30%, and the early postpartum period
SodiumHypernatraemiaHyponatraemia
Central catecholaminesDrugs that raise them: acute amphetamine or methamphetamine, cocaineDrugs that lower them; chronic amphetamine use
Central depressantsPremedication and sedatives, acute opioids (synergistic), α2 agonists, acute alcohol, lithium, lidocaine, neuraxial opioids
Other anaestheticsAdditive: nitrous oxide lowers the volatile concentration needed
CardiorespiratoryPaO2 below 5.1 kPa (38 mmHg); mean arterial pressure below 40 mmHg
OtherRed hair (melanocortin-1 receptor variants); ciclosporin; chronic opioid useCardiopulmonary bypass (inconsistent)

No change: sex, duration of anaesthesia, anaesthetic metabolism, PaCO2 from 2.0 to 12.7 kPa (15 to 95 mmHg), PaO2 above 5.1 kPa, mean arterial pressure above 40 mmHg, and hyperkalaemia or hypokalaemia.

In this patient: published MAC values are quoted for adults of about 40. At 50, with MAC falling about 6% per decade, the same end point needs roughly 6% less agent, before any opioid, sedative or temperature effect is added.

c

4 marks

Factors that dictate the speed of onset

Onset is the rate at which the partial pressure in the brain rises, and the brain follows the alveolus. So the question is what makes the alveolar fraction (FA) approach the inspired fraction (FI) quickly: delivery in, minus uptake out.

What earns the marks4 marks

The principleThe brain equilibrates with the alveolus; onset tracks the rise of FA/FI
Delivery to the alveolusInspired concentration (overpressure, concentration effect), fresh gas flow and circuit, alveolar ventilation, FRC
Uptake from the alveolusBlood:gas partition coefficient, cardiac output, alveolar to venous partial pressure difference
From blood to brainBrain:blood coefficient and cerebral blood flow
ModifiersSecond gas effect, shunt, airway irritability of the agent

Read the question: Describe” needs the direction and the reason for each factor. The one most often written backwards is solubility: a more soluble agent is slower, not faster, because blood keeps taking it away from the alveolus.

From vaporiser to brain, and what sets the speed at each step

Vaporiser and circuit
A high inspired concentration offsets uptake (overpressure). The circuit volume buffers the change; high fresh gas flow, 5 to 10 L/min, overcomes the buffer. Agent absorbed into rubber and plastic initially slows the rise.
Alveolus (FA/FI)
Raised by alveolar ventilation, and faster when FRC is small relative to ventilation. Lowered by uptake into pulmonary blood.

Uptake into blood, which slows the rise

Solubility
A high blood:gas coefficient means blood holds a large amount before its partial pressure rises.
Cardiac output
More pulmonary blood flow carries more agent away from the alveolus.
Venous return
Uptake falls as the vessel-rich tissues fill and mixed venous partial pressure rises.
Arterial blood
Equals the alveolar partial pressure unless a right-to-left shunt dilutes it.
Brain
Equilibrates with arterial blood in about three time constants, 5 to 15 minutes for the volatile agents. The brain:blood coefficient and cerebral blood flow govern this step.
FactorFaster onset whenWhy
Inspired concentrationHigherMore input offsets uptake; the higher the inspired concentration, the more rapidly FA approaches FI (the concentration effect)
Fresh gas flow and circuitHigh flow, small circuit volumeThe circuit is a reservoir to be filled before the patient receives the dialled concentration
Alveolar ventilationHigherMore agent delivered per minute; the effect is greatest for soluble agents. Spontaneous breathing gives negative feedback, as the agent depresses ventilation; controlled ventilation removes it
FRCSmall relative to ventilationLess gas to dilute the incoming agent. Alveolar ventilation to FRC is about 5:1 in neonates against 1.5:1 in adults, so induction is faster in neonates
Blood:gas partition coefficientLowLittle agent must dissolve before blood partial pressure rises. Anaemia lowers solubility (about 20% less at a haematocrit of 21%); a fatty meal raises it by about 20%
Cardiac outputLowLess agent carried away from the alveolus. Greatest effect with soluble agents; a low output state can produce an unexpectedly deep anaesthetic
Alveolar to venous differenceNarrowOnce vessel-rich tissues, 10% of body mass taking 75% of cardiac output, have equilibrated, less is taken up from the lung
Second gas effectGiven with high-concentration nitrous oxideRapid nitrous oxide uptake concentrates the volatile agent in a smaller alveolar volume and draws in more inspired gas
Right-to-left shuntAbsentShunted blood dilutes arterial partial pressure; this slows poorly soluble agents more than soluble ones
Airway irritabilityNon-pungent agentA pungent agent such as desflurane cannot be breathed at a high inspired concentration without coughing, breath-holding or laryngospasm
AgentBlood:gas coefficientOnset
Desflurane0.42Fastest
Sevoflurane0.69
Isoflurane1.46
Enflurane1.9
Halothane2.54Slowest
Connecting…
Account progress

Connecting your study progress…

Account & profile